Thyrotropin releasing hormone chloromethyl ketone structure

Thyrotropin releasing hormone chloromethyl ketone

(2S)-N-[(2S)-1-[(2S)-2-(2-chloroacetyl)pyrrolidin-1-yl]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide

Also Known As: Trh-cmk|Thyrotropin releasing hormone chloromethyl ketone|2-Pyrrolidinecarboxamide, N-(2-(2-(chloroacetyl)-1-pyrrolidinyl)-1-(1H-imidazol-4-ylmethyl)-2-oxoethyl)-5-oxo-, (2S-(2R*(R*(R*))))-|(2S)-N-[(2S)-1-[(2S)-2-(2-chloroacetyl)pyrrolidin-1-yl]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide|(2S)-N-[(2S)-1-[(2S)-2-(2-chloroacetyl)pyrrolidin-1-yl]-3-(3H-imidazol-4-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide|(2S)-N-[(2S)-1-[(2S)-2-(Chloroacetyl)pyrrolidin-1-yl]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-hydroxy-3,4-dihydro-2H-pyrrole-2-carboximidic acid|N-{1-[2-(Chloroacetyl)pyrrolidin-1-yl]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl}-5-hydroxy-3,4-dihydro-2H-pyrrole-2-carboximidic acid

CAS: 76819-95-9
Molecular Formula C17H22ClN5O4
Molecular Weight 395.13602 g/mol
LogP -1.0
Topological Polar Surface Area 124.0 Ų
Hydrogen Bond Donors 3
Hydrogen Bond Acceptors 5
Rotatable Bonds 7
Exact Mass 395.13602
Monoisotopic Mass 395.13602
Heavy Atoms 27
Complexity 616.0

Chemical Identifiers

CAS Number 76819-95-9
SMILES C1C[C@H](N(C1)C(=O)[C@H](CC2=CN=CN2)NC(=O)[C@@H]3CCC(=O)N3)C(=O)CCl
InChIKey IUYWTEQKCXPSLN-AVGNSLFASA-N

Product Overview

Thyrotropin releasing hormone chloromethyl ketone (CAS 76819-95-9), with molecular formula C17H22ClN5O4 and molecular weight 395.13602 g/mol. IUPAC: (2S)-N-[(2S)-1-[(2S)-2-(2-chloroacetyl)pyrrolidin-1-yl]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
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