Pivalopril structure

Pivalopril

2-[cyclopentyl-[3-(2,2-dimethylpropanoylsulfanyl)-2-methylpropanoyl]amino]acetic acid

Also Known As: Pivalopril|PIVOPRIL|Rhc-3659|Rhc 3659|Pivopril; RHC 3659(S)|2-[cyclopentyl-[3-(2,2-dimethylpropanoylsulfanyl)-2-methylpropanoyl]amino]acetic acid|N-cyclopentyl-N-(2-methyl-3-(pivaloylthio)propanoyl)glycine|N-Cyclopentyl-N-(3-((2,2-dimethyl-1-oxopropyl)thio)-2-methyl-1-oxypropyl)glycine|Glycine, N-cyclopentyl-N-(3-((2,2-dimethyl-1-oxopropyl)thio)-2-methyl-1-oxopropyl)-|{Cyclopentyl-[3-(2,2-dimethyl-propionylsulfanyl)-2-methyl-propionyl]-amino}-acetic acid|2-(N-cyclopentyl-2-{[(2,2-dimethylpropanoyl)sulfanyl]methyl}propanamido)acetic acid|N-Cyclopentyl-N-[2-methyl-3-[(2,2-dimethyl-1-oxopropyl)thio]-1-oxopropyl]glycine|(R)-{Cyclopentyl-[3-(2,2-dimethyl-propionylsulfanyl)-2-methyl-propionyl]-amino}-acetic acid|(S)-{Cyclopentyl-[3-(2,2-dimethyl-propionylsulfanyl)-2-methyl-propionyl]-amino}-acetic acid

CAS: 81045-50-3
Molecular Formula C16H27NO4S
Molecular Weight 329.16608 g/mol
LogP 2.9
Topological Polar Surface Area 100.0 Ų
Hydrogen Bond Donors 1
Hydrogen Bond Acceptors 5
Rotatable Bonds 8
Exact Mass 329.16608
Monoisotopic Mass 329.16608
Heavy Atoms 22
Complexity 424.0

Chemical Identifiers

CAS Number 81045-50-3
SMILES CC(CSC(=O)C(C)(C)C)C(=O)N(CC(=O)O)C1CCCC1
InChIKey XRKXJJYSKUIIEN-UHFFFAOYSA-N

Patent-Derived Application Labels

Derived from 8 IPC patent classification(s) across the SureChEMBL global patent database.

Agrochemicals (4 patents) Analytical Reagents (3 patents) Biotechnology (5 patents) Heterocyclic Building Blocks (39 patents) Organic Building Blocks (6 patents) Organometallic Reagents (2 patents) Peptides & Amino Acids (7 patents) Pharmaceutical Intermediates (51 patents)

Product Overview

Pivalopril (CAS 81045-50-3), with molecular formula C16H27NO4S and molecular weight 329.16608 g/mol. IUPAC: 2-[cyclopentyl-[3-(2,2-dimethylpropanoylsulfanyl)-2-methylpropanoyl]amino]acetic acid.

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Safety Data Sheet (MSDS / SDS) View the Laboratory Chemical Safety Summary (LCSS) on PubChem — includes GHS classifications, hazard statements, first aid measures, and handling precautions.
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